Examinant per Autoria "Stepniewski, Tomasz Maciej, 1988-"
Resultats per pàgina
Opcions d'ordenació
Ítem Accés Obert A molecular sensor for cholesterol in the human serotonin 1A receptor(American Association for the Advancement of Science (AAAS), 2021) Kumar, G Aditya; Sarkar, Parijat; Stepniewski, Tomasz Maciej, 1988-; Jafurulla, Md; Singh, Shishu Pal; Selent, Jana; Chattopadhyay, Amitabha
Ítem Accés Obert Allosteric modulation of GPCR-induced β-arrestin trafficking and signaling by a synthetic intrabody(Nature Research, 2022) Baidya, Mithu; Chaturvedi, Madhu; Dwivedi, Hemlata; Ranjan, Ashutosh; Devost, Dominic; Namkung, Yoon; Stepniewski, Tomasz Maciej, 1988-; Pandey, Shubhi; Baruah, Minakshi; Panigrahi, Bhanupriya; Sarma, Parishmita; Yadav, Manish K.; Maharana, Jagannath; Banerjee, Ramanuj; Kawakami, Kouki; Inoue, Asuka; Selent, Jana; Laporte, Stéphane A.; Hébert, Terence E.; Shukla, Arun K.
Ítem Accés Obert Discovery of a dual Ras and ARF6 inhibitor from a GPCR endocytosis screen(Nature Research, 2021) Giubilaro, Jenna; Schuetz, Doris A.; Stepniewski, Tomasz Maciej, 1988-; Namkung, Yoon; Khoury, Etienne; Lara Márquez, Mónica; Campbell, Shirley; Beautrait, Alexandre; Armando, Sylvain; Radresa, Olivier; Duchaine, Jean; Lamarche Vane, Nathalie; Claing, Audrey; Selent, Jana; Bouvier, Michel; Marinier, Anne; Laporte, Stéphane A.
Ítem Accés Obert Distinct phosphorylation sites in a prototypical GPCR differently orchestrate β-arrestin interaction, trafficking, and signaling(American Association for the Advancement of Science (AAAS), 2020) Dwivedi, Hemlata; Chaturvedi, Madhu; Baidya, Mithu; Stepniewski, Tomasz Maciej, 1988-; Pandey, Shubhi; Maharana, Jagannath; Srivastava, Ashish; Caengprasath, Natarin; Hanyaloglu, Aylin C.; Selent, Jana; Shukla, Arun K.
Ítem Accés Obert Do they make a good match? Molecular dynamics studies on CALB-catalyzed esterification of 3-phenylpropionic and cinnamic acids(Elsevier, 2023) Zieniuk, Bartlomiej; Stepniewski, Tomasz Maciej, 1988-; Fabiszewska, Agata
Ítem Accés Obert Dopamine D 2 receptor agonist binding kinetics-role of a conserved serine residue(MDPI, 2021) Ågren, Richard; Stepniewski, Tomasz Maciej, 1988-; Zeberg, Hugo; Selent, Jana; Sahlholm, Kristoffer
Ítem Accés Obert Entrectinib-A SARS-CoV-2 inhibitor in Human Lung Tissue (HLT) cells(MDPI, 2021) Peralta-Garcia, Alejandro; Torrens Fontanals, Mariona; Stepniewski, Tomasz Maciej, 1988-; Grau-Expósito, Judith; Perea, David; Ayinampudi, Vikram; Waldhoer, Maria; Zimmermann, Mirjam; Buzón, María J.; Genescà, Meritxell; Selent, Jana
Ítem Accés Obert G protein-specific mechanisms in the serotonin 5-HT2A receptor regulate psychosis-related effects and memory deficits(Nature Research, 2024) Kossatz de Mello, Elk, 1977-; Diez Alarcia, Rebeca; Gaitonde, Supriya A.; Ramon Duaso, Carla, 1987-; Stepniewski, Tomasz Maciej, 1988-; Aranda García, David; Muneta Arrate, Itziar; Tepaz, Elodie; Saen-Oon, Suwipa; Soliva, Robert; Shahraki, Aida; Moreira, David; Brea, José; Loza, María I.; Torre Fornell, Rafael de la; Kolb, Peter; Bouvier, Michel; Meana, J. Javier; Robledo, Patricia, 1958-; Selent, Jana
Ítem Accés Obert How do molecular dynamics data complement static structural data of GPCRs(MDPI, 2020) Torrens Fontanals, Mariona; Stepniewski, Tomasz Maciej, 1988-; Aranda García, David; Morales Pastor, Adrián; Medel Lacruz, Brian; Selent, Jana
Ítem Accés Obert Ligand entry pathways control the chemical space recognized by GPR183(Royal Society of Chemistry, 2023) Kjaer, Viktoria Madeline Skovgaard; Stepniewski, Tomasz Maciej, 1988-; Medel Lacruz, Brian; Reinmuth, Lisa; Ciba, Marija; Rexen Ulven, Elisabeth; Bonomi, Massimiliano; Selent, Jana; Rosenkilde, Mette Marie
Ítem Accés Obert Ligand with two modes of interaction with the dopamine D2 receptor-an induced-fit mechanism of insurmountable antagonism(American Chemical Society (ACS), 2020) Ågren, Richard; Zeberg, Hugo; Stepniewski, Tomasz Maciej, 1988-; Free, R. Benjamin; Reilly, Sean W.; Luedtke, Robert R.; Århem, Peter; Ciruela, Francisco; Sibley, David R.; Mach, Robert H.; Selent, Jana; Nilsson, Johanna; Sahlholm, Kristoffer
Ítem Accés Obert Mechanistic insights into dopaminergic and serotonergic neurotransmission - concerted interactions with helices 5 and 6 drive the functional outcome(Royal Society of Chemistry, 2021) Stepniewski, Tomasz Maciej, 1988-; Mancini, Arturo; Ågren, Richard; Torrens Fontanals, Mariona; Semache, Meriem; Bouvier, Michel; Sahlholm, Kristoffer; Breton, Billy; Selent, Jana
Ítem Accés Obert Oxazoline scaffold in synthesis of benzosiloxaboroles and related ring-expanded heterocycles: diverse reactivity, structural peculiarities and antimicrobial activity(Royal Society of Chemistry, 2022) Krajewska, Joanna; Nowicki, Krzysztof; Durka, Krzysztof; Marek-Urban, Paulina H.; Wińska, Patrycja; Stepniewski, Tomasz Maciej, 1988-; Woźniak, Krzysztof; Laudy, Agnieszka E.; Luliński, Sergiusz
Ítem Accés Obert Plasma membrane preassociation drives β-arrestin coupling to receptors and activation(Elsevier, 2023) Grimes, Jak; Koszegi, Zsombor; Lanoiselée, Yann; Miljus, Tamara; O'Brien, Shannon L.; Stepniewski, Tomasz Maciej, 1988-; Medel Lacruz, Brian; Baidya, Mithu; Makarova, Maria; Mistry, Ravi; Goulding, Joëlle; Drube, Julia; Hoffmann, Carsten; Owen, Dylan M.; Shukla, Arun K.; Selent, Jana; Hill, Stephen J.; Calebiro, Davide
Ítem Accés Obert Relevance of G protein-coupled receptor (GPCR) dynamics for receptor activation, signalling bias and allosteric modulation(Wiley, 2024) Lopez-Balastegui, Marta; Stepniewski, Tomasz Maciej, 1988-; Kogut-Günthel, Małgorzata M.; Di Pizio, Antonella; Rosenkilde, Mette Marie; Mao, Jiafei; Selent, Jana